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Assay Detail

CHEMBL4715266

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of 5'-FAM/3'-DAB-labeled UGUCGGGUAGCUUAUCAGACUGAUGUUGACUGUUGAAUCUCAUGGCAACACCAGUCGAUGGGCUGUCUGACA pre-miRNA-21 (unknown origin) biogenesis preincubated for 30 mins followed by MCF7 cell lysate addition and measured after 1 hr by fluorescence based assay
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Not specified
Confidence 3 — Cell-line / Tissue
Curated By Autocuration

Target

microRNA 21 (CHEMBL1615322)
Type NUCLEIC-ACID
Organism Homo sapiens

Publication

Design and Implementation of Synthetic RNA Binders for the Inhibition of miR-21 Biogenesis.
Maucort C,Vo DD,Aouad S,Charrat C,Azoulay S,Di Giorgio A,Duca M
ACS Med Chem Lett (2021) 12 : 899 -906
PubMed 34141067 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 5.51 5.51

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL4762976 1 5.51

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL4762976 IC50 = 3100.0 nM 5.51