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Assay Detail

CHEMBL4717285

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Binding
Binding affinity to actin (unknown origin) assessed as dissociation constant for actin-compound-tubulin heterodimer complex at 25 degreeC
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Confidence 0 — Uncurated / Unknown
Curated By Autocuration

Target

Unchecked (CHEMBL612545)
Type UNCHECKED

Publication

Analysis of the aplyronine A-induced protein-protein interaction between actin and tubulin by surface plasmon resonance.
Hirayama Y,Yamagishi K,Suzuki T,Kawagishi H,Kita M,Kigoshi H
Bioorg Med Chem (2016) 24 : 2809 -2814
PubMed 27161875 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Kd 1 5.74 5.74

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL412190 APLYRONINE A 1 5.74

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL412190 APLYRONINE A Kd = 1840.0 nM 5.74