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Assay Detail

CHEMBL4723487

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of envelope protein in Murine hepatitis virus A59 infected in mouse L929 cells assessed as reduction in viral replication incubated for 24 hrs by crystal violet staining based plaque reduction assay
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Murine hepatitis virus
Cell Type L929
Confidence 0 — Uncurated / Unknown
Curated By Autocuration

Target

Unchecked (CHEMBL612545)
Type UNCHECKED

Publication

Druggable targets from coronaviruses for designing new antiviral drugs.
Silva LR,da Silva Santos-Júnior PF,de Andrade Brandão J,Anderson L,Bassi ÊJ,Xavier de Araújo-Júnior J,Cardoso SH,da Silva-Júnior EF
Bioorg Med Chem (2020) 28 : 115745 -115745
PubMed 33007557 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 1 5.41 5.41

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL501701 N,N-HEXAMETHYLENEAMILORIDE 1 5.41

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL501701 N,N-HEXAMETHYLENEAMILORIDE EC50 = 3910.0 nM 5.41