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Assay Detail

CHEMBL4723495

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of N-terminus hexa-histidine tagged-SARS-coV guanine-N7 methyltransferase expressed in Escherichia coli using GpppAUAU RNA as substrate incubated for 30 mins by liquid scintillation counting method
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Severe acute respiratory syndrome-related coronavirus
Confidence 0 — Uncurated / Unknown
Curated By Autocuration

Target

Unchecked (CHEMBL612545)
Type UNCHECKED

Publication

Druggable targets from coronaviruses for designing new antiviral drugs.
Silva LR,da Silva Santos-Júnior PF,de Andrade Brandão J,Anderson L,Bassi ÊJ,Xavier de Araújo-Júnior J,Cardoso SH,da Silva-Júnior EF
Bioorg Med Chem (2020) 28 : 115745 -115745
PubMed 33007557 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 7.72 7.72

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL6246 ELLAGIC ACID 2.0 1 7.72

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL6246 ELLAGIC ACID IC50 = 19.0 nM 7.72