Assay Detail
Binding
CHEMBL4723780
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Binding affinity to human CAMKK1 assessed as displacement of immobilized ligand by KINOMEscan scanMAX assay relative to control
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Calcium/calmodulin-dependent protein kinase kinase 1 (CHEMBL5256) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
A Chemical Probe for Dark Kinase STK17B Derives Its Potency and High Selectivity through a Unique P-Loop Conformation.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Kd | 1 | 7.31 | 7.31 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4752776 | — | — | 1 | 7.31 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4752776 | — | Kd | = | 49.0 | nM | 7.31 |