Assay Detail
Binding
CHEMBL4730904
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Binding affinity to NF-kappaB RelA (unknown origin) by SPR analysis
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Gibberellin JRA-003: A Selective Inhibitor of Nuclear Translocation of IKKα.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Kd | 2 | 5.05 | 5.20 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL2359602 | — | — | 1 | 5.20 |
| CHEMBL1232952 | GIBBERELLIN A3 | — | 1 | 4.89 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL2359602 | — | Kd | = | 6340.0 | nM | 5.20 |
| CHEMBL1232952 | GIBBERELLIN A3 | Kd | = | 13000.0 | nM | 4.89 |