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Assay Detail

CHEMBL4732474

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Cytotoxicity against mouse B16-F10 cells assessed as reduction in cell viability measured after 72 hrs by MTT assay
7
Total Activities
7
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Mus musculus
Cell Type B16-F10
Confidence 1 — Organism
Curated By Autocuration

Target

B16-F10 (CHEMBL612656)
Type CELL-LINE
Organism Mus musculus

Publication

Benzimidazole-1,2,3-triazole hybrid molecules: synthesis and study of their interaction with G-quadruplex DNA
Singu, Padma S., Chilakamarthi, Ushasri, Mahadik, Namita S., Keerti, Bhamidipati, Valipenta, Narasimhulu, Mokale, Santosh N., Nagesh, Narayana, Kumbhare, Ravindra M.
RSC Med Chem (2021) 12 : 416 -429
PubMed 34046624 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 7 4.12 4.25

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL4764858 1 4.25
CHEMBL65606 TMPYP4 1 4.11
CHEMBL4786759 1 4.07
CHEMBL4750911 1 4.04
CHEMBL4759761 1 -
CHEMBL4753593 1 -
CHEMBL4781867 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL4764858 IC50 = 56790.0 nM 4.25
CHEMBL65606 TMPYP4 IC50 = 77010.0 nM 4.11
CHEMBL4786759 IC50 = 84680.0 nM 4.07
CHEMBL4750911 IC50 = 90500.0 nM 4.04
CHEMBL4759761 IC50 = 203000.0 nM -
CHEMBL4753593 IC50 = 135000.0 nM -
CHEMBL4781867 IC50 = 103000.0 nM -