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Assay Detail

CHEMBL4732475

Review assay metadata, readout intent, target linkage, and publication context from the same page.

ADMET
Cytotoxicity against human CHO-K1 cells assessed as reduction in cell viability measured after 72 hrs by MTT assay
7
Total Activities
7
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type ADMET
Organism Cricetulus griseus
Cell Type CHO-K1
Confidence 1 — Organism
Curated By Autocuration

Target

CHO-K1 (CHEMBL614031)
Type CELL-LINE
Organism Cricetulus griseus

Publication

Benzimidazole-1,2,3-triazole hybrid molecules: synthesis and study of their interaction with G-quadruplex DNA
Singu, Padma S., Chilakamarthi, Ushasri, Mahadik, Namita S., Keerti, Bhamidipati, Valipenta, Narasimhulu, Mokale, Santosh N., Nagesh, Narayana, Kumbhare, Ravindra M.
RSC Med Chem (2021) 12 : 416 -429
PubMed 34046624 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 7 4.19 4.25

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL4764858 1 4.25
CHEMBL4781867 1 4.21
CHEMBL65606 TMPYP4 1 4.21
CHEMBL4786759 1 4.20
CHEMBL4750911 1 4.07
CHEMBL4759761 1 -
CHEMBL4753593 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL4764858 IC50 = 56100.0 nM 4.25
CHEMBL4781867 IC50 = 62210.0 nM 4.21
CHEMBL65606 TMPYP4 IC50 = 61400.0 nM 4.21
CHEMBL4786759 IC50 = 62900.0 nM 4.20
CHEMBL4750911 IC50 = 85050.0 nM 4.07
CHEMBL4759761 IC50 = 100380.0 nM -
CHEMBL4753593 IC50 = 114670.0 nM -