Assay Detail
ADMET
CHEMBL4733261
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Cytotoxicity against human peripheral blood lymphocytes assessed as cell viability after 72 hrs by luminescent assay
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | ADMET |
| Organism | Homo sapiens |
| Cell Type | Lymphocyte |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Cyclic bridged analogs of isoCA-4: Design, synthesis and biological evaluation.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 6.86 | 6.86 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4798567 | — | — | 1 | 6.86 |
| CHEMBL498271 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4798567 | — | IC50 | = | 137.0 | nM | 6.86 |
| CHEMBL498271 | — | IC50 | > | 10.0 | nM | - |