Assay Detail
Functional
CHEMBL4735356
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Antiproliferative activity against human Pfeiffer cells incubated for 10 days by cellTiter-glo luminesence method
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | Pfeiffer |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Small Molecule Approaches for Targeting the Polycomb Repressive Complex 2 (PRC2) in Cancer.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 1 | 7.16 | 7.16 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4104741 | — | — | 1 | 7.16 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4104741 | — | IC50 | = | 69.0 | nM | 7.16 |