Assay Detail
Binding
CHEMBL4738703
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of SARS CoV papain-like protease using Arg-Leu-Arg-Gly-Gly-AMC as substrate by fluorescence method
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Severe acute respiratory syndrome-related coronavirus |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Protease targeted COVID-19 drug discovery: What we have learned from the past SARS-CoV inhibitors?
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 1 | 5.39 | 5.39 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL464274 | DEHYDROHIRSUTANONOL | — | 1 | 5.39 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL464274 | DEHYDROHIRSUTANONOL | IC50 | = | 4100.0 | nM | 5.39 |