Assay Detail
Functional
CHEMBL4739787
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Antiproliferative activity against human HAP1 cells harboring CDK12 C1039S/CDK13 C1017S double mutant measured after 72 hrs by CellTiter-Glo Luminescent Cell Viability Assay
15
Total Activities
15
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | HAP1 |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Inhibitors of cyclin-dependent kinases
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 15 | 6.04 | 6.51 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4781539 | — | — | 1 | 6.51 |
| CHEMBL4788401 | — | — | 1 | 6.23 |
| CHEMBL4777841 | — | — | 1 | 6.21 |
| CHEMBL4751989 | — | — | 1 | 6.03 |
| CHEMBL4756935 | — | — | 1 | 5.96 |
| CHEMBL4636175 | — | — | 1 | 5.30 |
| CHEMBL4777761 | — | — | 1 | - |
| CHEMBL4790868 | — | — | 1 | - |
| CHEMBL4749580 | — | — | 1 | - |
| CHEMBL4763994 | — | — | 1 | - |
| CHEMBL4743840 | — | — | 1 | - |
| CHEMBL4763202 | — | — | 1 | - |
| CHEMBL4794338 | — | — | 1 | - |
| CHEMBL4764719 | — | — | 1 | - |
| CHEMBL4781334 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4781539 | — | IC50 | = | 308.0 | nM | 6.51 |
| CHEMBL4788401 | — | IC50 | = | 591.0 | nM | 6.23 |
| CHEMBL4777841 | — | IC50 | = | 618.0 | nM | 6.21 |
| CHEMBL4751989 | — | IC50 | = | 944.0 | nM | 6.03 |
| CHEMBL4756935 | — | IC50 | = | 1096.0 | nM | 5.96 |
| CHEMBL4636175 | — | IC50 | = | 4960.0 | nM | 5.30 |
| CHEMBL4777761 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL4790868 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL4749580 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL4763994 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL4743840 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL4763202 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL4794338 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL4764719 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL4781334 | — | IC50 | > | 10000.0 | nM | - |