Assay Detail
Binding
CHEMBL4739818
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of recombinant CLK2 (unknown origin) using Ser/Thr 6 peptide as substrate incubated for 1 hr in presence of ATP by FRET assay
641
Total Activities
641
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Dual specificity protein kinase CLK2 (CHEMBL4225) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
Methods of treating cartilage disorders through inhibition of clk and dyrk
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 641 | 8.35 | 9.00 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4797346 | — | — | 1 | 9.00 |
| CHEMBL4748995 | — | — | 1 | 9.00 |
| CHEMBL4794727 | — | — | 1 | 9.00 |
| CHEMBL4756030 | — | — | 1 | 9.00 |
| CHEMBL4782319 | — | — | 1 | 9.00 |
| CHEMBL4788275 | — | — | 1 | 9.00 |
| CHEMBL4752625 | — | — | 1 | 9.00 |
| CHEMBL4779592 | — | — | 1 | 9.00 |
| CHEMBL4742725 | — | — | 1 | 9.00 |
| CHEMBL4800084 | — | — | 1 | 9.00 |
| CHEMBL4776499 | — | — | 1 | 9.00 |
| CHEMBL4754606 | — | — | 1 | 9.00 |
| CHEMBL4761354 | — | — | 1 | 9.00 |
| CHEMBL4795039 | — | — | 1 | 9.00 |
| CHEMBL4800437 | — | — | 1 | 9.00 |
| CHEMBL4743901 | — | — | 1 | 9.00 |
| CHEMBL4788156 | — | — | 1 | 9.00 |
| CHEMBL4790477 | — | — | 1 | 9.00 |
| CHEMBL4746176 | — | — | 1 | 9.00 |
| CHEMBL4778412 | — | — | 1 | 9.00 |
| CHEMBL4760183 | — | — | 1 | 9.00 |
| CHEMBL4745311 | — | — | 1 | 9.00 |
| CHEMBL4742870 | — | — | 1 | 9.00 |
| CHEMBL4750147 | — | — | 1 | 9.00 |
| CHEMBL4785637 | — | — | 1 | 9.00 |
| CHEMBL4761714 | — | — | 1 | 9.00 |
| CHEMBL4791039 | — | — | 1 | 9.00 |
| CHEMBL4741792 | — | — | 1 | 9.00 |
| CHEMBL4755807 | — | — | 1 | 9.00 |
| CHEMBL4788267 | — | — | 1 | 9.00 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4794020 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL4779592 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL4752625 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL4762097 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL4755887 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL4747934 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL4747908 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL4756183 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL4777667 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL4744357 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL4744452 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL4778878 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL4751049 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL4748484 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL4756656 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL4741843 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL4796085 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL4786934 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL4782319 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL4756030 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL4794727 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL4800211 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL4748995 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL4743856 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL4761662 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL4795039 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL4745311 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL4788493 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL4783753 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL4745861 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL4760183 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL4778412 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL4746176 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL4790477 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL4788156 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL4797346 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL4800437 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL4744439 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL4788275 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL4761354 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL4750400 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL4754511 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL4784318 | CIRTUVIVINT | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL4754606 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL4776499 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL4757954 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL4800084 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL4746707 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL4778742 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL4742725 | — | EC50 | = | 1.0 | nM | 9.00 |