Assay Detail
Binding
CHEMBL4767576
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Inhibition of mouse GTA 3 receptor
8
Total Activities
8
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Mus musculus |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Novel mouse GABA uptake inhibitors with enhanced inhibitory activity toward mGAT3/4 and their effect on pain threshold in mice.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 8 | 4.95 | 5.29 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3289575 | — | — | 1 | 5.29 |
| CHEMBL419823 | — | — | 1 | 5.29 |
| CHEMBL96 | GAMMA-AMINOBUTYRIC ACID | 1.0 | 1 | 5.15 |
| CHEMBL4779064 | — | — | 1 | 4.85 |
| CHEMBL297569 | BETA-ALANINE | — | 1 | 4.18 |
| CHEMBL4566905 | — | — | 1 | - |
| CHEMBL4793097 | — | — | 1 | - |
| CHEMBL4789121 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3289575 | — | IC50 | = | 5128.61 | nM | 5.29 |
| CHEMBL419823 | — | IC50 | = | 5128.61 | nM | 5.29 |
| CHEMBL96 | GAMMA-AMINOBUTYRIC ACID | IC50 | = | 7079.46 | nM | 5.15 |
| CHEMBL4779064 | — | IC50 | = | 14125.38 | nM | 4.85 |
| CHEMBL297569 | BETA-ALANINE | IC50 | = | 66069.34 | nM | 4.18 |
| CHEMBL4566905 | — | IC50 | = | 181970.09 | nM | - |
| CHEMBL4793097 | — | IC50 | = | 301995.17 | nM | - |
| CHEMBL4789121 | — | IC50 | = | 301995.17 | nM | - |