Assay Detail
Binding
CHEMBL4771534
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of HDAC11 (unknown origin)
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Thirty Years of HDAC Inhibitors: 2020 Insight and Hindsight.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 7.96 | 9.52 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL343448 | ROMIDEPSIN | 4.0 | 1 | 9.52 |
| CHEMBL3621988 | TUCIDINOSTAT | 3.0 | 1 | 6.40 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL343448 | ROMIDEPSIN | IC50 | = | 0.3 | nM | 9.52 |
| CHEMBL3621988 | TUCIDINOSTAT | IC50 | = | 400.0 | nM | 6.40 |