Assay Detail
Binding
CHEMBL4772219
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Displacement of [125I][Tyr1]-NPFF from NPFF receptor in rat spinal cord membranes by Cheng-Prusoff analysis
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Rattus norvegicus |
| Tissue | Spinal cord |
| Subcellular | Membrane |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Neuropeptide FF and Its Receptors: Therapeutic Applications and Ligand Development.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 3 | 9.43 | 9.70 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL269186 | — | — | 1 | 9.70 |
| CHEMBL429731 | — | — | 1 | 9.68 |
| CHEMBL407343 | — | — | 1 | 8.92 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL269186 | — | Ki | = | 0.2 | nM | 9.70 |
| CHEMBL429731 | — | Ki | = | 0.21 | nM | 9.68 |
| CHEMBL407343 | — | Ki | = | 1.2 | nM | 8.92 |