Assay Detail
Binding
CHEMBL4772225
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Displacement of [125I]YVP from human NPFFR1 expressed in CHO cells by gamma-counter method
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Cell Type | CHO |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Neuropeptide FF and Its Receptors: Therapeutic Applications and Ligand Development.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 2 | 8.89 | 9.23 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL2165920 | — | — | 1 | 9.23 |
| CHEMBL4460742 | — | — | 1 | 8.54 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL2165920 | — | Ki | = | 0.59 | nM | 9.23 |
| CHEMBL4460742 | — | Ki | = | 2.9 | nM | 8.54 |