Assay Detail
Binding
CHEMBL4772233
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Displacement of [125I]Tyr-NPFF from human NPFFR2 expressed in green monkey Cos-1 cells
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Cell Type | COS-1 |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Neuropeptide FF and Its Receptors: Therapeutic Applications and Ligand Development.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 2 | 6.73 | 7.12 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1672380 | — | — | 1 | 7.12 |
| CHEMBL2440929 | — | — | 1 | 6.34 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1672380 | — | Ki | = | 75.0 | nM | 7.12 |
| CHEMBL2440929 | — | Ki | = | 461.0 | nM | 6.34 |