Assay Detail
Binding
CHEMBL4772272
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Agonist activity at NPFFR2 (unknown origin) expressed in mouse NIH3T3 cells by receptor selection and amplification technology assay
4
Total Activities
4
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Cell Type | NIH3T3 |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Neuropeptide FF and Its Receptors: Therapeutic Applications and Ligand Development.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 4 | 6.40 | 7.00 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4785076 | — | — | 1 | 7.00 |
| CHEMBL4794542 | — | — | 1 | 6.40 |
| CHEMBL3982697 | — | — | 1 | 6.10 |
| CHEMBL4784123 | — | — | 1 | 6.10 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4785076 | — | EC50 | = | 100.0 | nM | 7.00 |
| CHEMBL4794542 | — | EC50 | = | 398.11 | nM | 6.40 |
| CHEMBL3982697 | — | EC50 | = | 794.33 | nM | 6.10 |
| CHEMBL4784123 | — | EC50 | = | 794.33 | nM | 6.10 |