Assay Detail
Functional
CHEMBL4772274
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Agonist activity at NPFFR1 (unknown origin) expressed in HEK293T cells harboring EP2 incubated for 15 mins by cAMP assay
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | HEK293T |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Neuropeptide FF and Its Receptors: Therapeutic Applications and Ligand Development.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 3 | 5.40 | 5.90 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4785076 | — | — | 1 | 5.90 |
| CHEMBL4794542 | — | — | 1 | 5.50 |
| CHEMBL4784123 | — | — | 1 | 4.80 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4785076 | — | EC50 | = | 1258.93 | nM | 5.90 |
| CHEMBL4794542 | — | EC50 | = | 3162.28 | nM | 5.50 |
| CHEMBL4784123 | — | EC50 | = | 15848.93 | nM | 4.80 |