Assay Detail
Binding
CHEMBL4772710
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Inhibition of human recombinant S100P/RAGE interaction incubated for 1 hr and measured at 100 nM by ELISA based binding assay
16
Total Activities
16
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Discovery of novel small molecule inhibitors of S100P with in vitro anti-metastatic effects on pancreatic cancer cells.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 16 | 8.18 | 9.32 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4797038 | — | — | 1 | 9.32 |
| CHEMBL4791219 | — | — | 1 | 9.29 |
| CHEMBL4776927 | — | — | 1 | 9.26 |
| CHEMBL4789650 | — | — | 1 | 9.22 |
| CHEMBL4778482 | — | — | 1 | 9.10 |
| CHEMBL4791820 | — | — | 1 | 8.89 |
| CHEMBL4778710 | — | — | 1 | 8.38 |
| CHEMBL4793118 | — | — | 1 | 8.16 |
| CHEMBL4784354 | — | — | 1 | 8.11 |
| CHEMBL4791308 | — | — | 1 | 7.86 |
| CHEMBL3191438 | — | — | 1 | 7.72 |
| CHEMBL4794659 | — | — | 1 | 7.64 |
| CHEMBL4784003 | — | — | 1 | 7.37 |
| CHEMBL4521239 | — | — | 1 | 7.11 |
| CHEMBL4799826 | — | — | 1 | 6.90 |
| CHEMBL1577938 | — | — | 1 | 6.58 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4797038 | — | IC50 | = | 0.482 | nM | 9.32 |
| CHEMBL4791219 | — | IC50 | = | 0.514 | nM | 9.29 |
| CHEMBL4776927 | — | IC50 | = | 0.555 | nM | 9.26 |
| CHEMBL4789650 | — | IC50 | = | 0.6 | nM | 9.22 |
| CHEMBL4778482 | — | IC50 | = | 0.796 | nM | 9.10 |
| CHEMBL4791820 | — | IC50 | = | 1.3 | nM | 8.89 |
| CHEMBL4778710 | — | IC50 | = | 4.15 | nM | 8.38 |
| CHEMBL4793118 | — | IC50 | = | 6.89 | nM | 8.16 |
| CHEMBL4784354 | — | IC50 | = | 7.7 | nM | 8.11 |
| CHEMBL4791308 | — | IC50 | = | 13.9 | nM | 7.86 |
| CHEMBL3191438 | — | IC50 | = | 19.0 | nM | 7.72 |
| CHEMBL4794659 | — | IC50 | = | 22.7 | nM | 7.64 |
| CHEMBL4784003 | — | IC50 | = | 42.6 | nM | 7.37 |
| CHEMBL4521239 | — | IC50 | = | 77.0 | nM | 7.11 |
| CHEMBL4799826 | — | IC50 | = | 126.0 | nM | 6.90 |
| CHEMBL1577938 | — | IC50 | = | 264.0 | nM | 6.58 |