Assay Detail
Functional
CHEMBL4807540
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Cytotoxicity against human NCI-H1299 cells assessed as inhibition of cell growth after 72 hrs by ATPlite assay
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | NCI-H1299 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Nek6 kinase inhibitors useful for the treatment of solid tumors
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 4.06 | 4.06 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4875865 | — | — | 1 | 4.06 |
| CHEMBL4862849 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4875865 | — | IC50 | = | 87800.0 | nM | 4.06 |
| CHEMBL4862849 | — | IC50 | > | 100000.0 | nM | - |