Assay Detail
Binding
CHEMBL4807555
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of human PIK3C2A using phosphatidylinositol as substrate and 10 uM ATP after 1 hr by TR-FRET based Adapta universal kinase assay
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Phosphatidylinositol 4-phosphate 3-kinase C2 domain-containing subunit alpha (CHEMBL1075102) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
Methods for treating centronuclear myopathy
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 1 | 8.02 | 8.02 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4869265 | — | — | 1 | 8.02 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4869265 | — | IC50 | = | 9.57 | nM | 8.02 |