Assay Detail
Binding
CHEMBL4813153
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of human Nav1.5 VSD4 R1628A mutant by automated voltage clamp electrophysiology
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Identification of aryl sulfonamides as novel and potent inhibitors of Na<sub>V</sub>1.5.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 1 | 6.09 | 6.09 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4859414 | — | — | 1 | 6.09 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4859414 | — | IC50 | = | 820.0 | nM | 6.09 |