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Assay Detail

CHEMBL4813249

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Noncompetitive inhibition of mushroom tyrosinase assessed as dissociation constant using L-DOPA as substrate by Lineweaver-Burk plot analysis
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Agaricus bisporus
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Tyrosinase (CHEMBL3318)
Type SINGLE PROTEIN
Organism Agaricus bisporus

Publication

Novel 1,3,4-oxadiazole compounds inhibit the tyrosinase and melanin level: Synthesis, in-vitro, and in-silico studies.
Vanjare BD, Choi NG, Mahajan PG, Raza H, Hassan M, Han Y, Yu SM, Kim SJ, Seo SY, Lee KH.
Bioorg Med Chem (2021) 41 : 116222 -116222
PubMed 34058664 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 1 8.51 8.51

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL1481541 1 8.51

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL1481541 Ki = 3.1 nM 8.51