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Assay Detail

CHEMBL4816212

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Functional
Inhibition of colony formation in human OVCAR-3 cells overexpressing G6PD incubated for 14 days by crystal violet staining based assay
2
Total Activities
1
Compounds Tested
2
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Homo sapiens
Cell Type OVCAR-3
Confidence 1 — Organism
Curated By Autocuration

Target

OVCAR-3 (CHEMBL614213)
Type CELL-LINE
Organism Homo sapiens

Publication

Discovery and characterization of a novel glucose-6-phosphate dehydrogenase (G6PD) inhibitor via high-throughput screening.
Luo Z, Du D, Liu Y, Lu T, Liu L, Jiang H, Chen K, Shan C, Luo C.
Bioorg Med Chem Lett (2021) 40 : 127905 -127905
PubMed 33689874 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 1 4.97 4.97
Inhibition 1 - -

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL97453 WEDELOLACTONE 2 4.97

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL97453 WEDELOLACTONE EC50 = 10640.0 nM 4.97
CHEMBL97453 WEDELOLACTONE Inhibition - % -