Assay Detail
Binding
CHEMBL4817199
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Inhibition of MurF (unknown origin)
7
Total Activities
7
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Not specified |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Mur ligases inhibitors with azastilbene scaffold: Expanding the structure-activity relationship.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 7 | 4.42 | 4.77 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4869060 | — | — | 1 | 4.77 |
| CHEMBL4877363 | — | — | 1 | 4.51 |
| CHEMBL373576 | — | — | 1 | 4.23 |
| CHEMBL4863582 | — | — | 1 | 4.15 |
| CHEMBL4879187 | — | — | 1 | - |
| CHEMBL4855039 | — | — | 1 | - |
| CHEMBL4875957 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4869060 | — | IC50 | = | 17000.0 | nM | 4.77 |
| CHEMBL4877363 | — | IC50 | = | 31000.0 | nM | 4.51 |
| CHEMBL373576 | — | IC50 | = | 59000.0 | nM | 4.23 |
| CHEMBL4863582 | — | IC50 | = | 71000.0 | nM | 4.15 |
| CHEMBL4879187 | — | IC50 | = | 109000.0 | nM | - |
| CHEMBL4855039 | — | IC50 | = | 144000.0 | nM | - |
| CHEMBL4875957 | — | IC50 | = | 201000.0 | nM | - |