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Assay Detail

CHEMBL4819448

Review assay metadata, readout intent, target linkage, and publication context from the same page.

ADMET
Cytotoxicity against human HL7702 cells incubated for 48 hrs by MTT assay
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type ADMET
Organism Homo sapiens
Cell Type L02
Confidence 1 — Organism
Curated By Autocuration

Target

L02 (CHEMBL4296457)
Type CELL-LINE
Organism Homo sapiens

Publication

Recent advances of podophyllotoxin/epipodophyllotoxin hybrids in anticancer activity, mode of action, and structure-activity relationship: An update (2010-2020).
Xiao J, Gao M, Sun Z, Diao Q, Wang P, Gao F.
Eur J Med Chem (2020) 208 : 112830 -112830
PubMed 32992133 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 3 6.14 6.52

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL4847670 1 6.52
CHEMBL4869119 1 6.52
CHEMBL61 PODOFILOX 4.0 1 5.37

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL4847670 IC50 = 300.0 nM 6.52
CHEMBL4869119 IC50 = 300.0 nM 6.52
CHEMBL61 PODOFILOX IC50 = 4310.0 nM 5.37