Assay Detail
Binding
CHEMBL4826966
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Displacement of [3H]2-BFI from imidazoline I2 receptor high affinity site in Swiss mouse brain cerebral cortex membrane measured after 30 mins by liquid scintillation counting spectrometry
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Mus musculus |
| Tissue | Cortex |
| Subcellular | Membrane |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Benzofuranyl-2-imidazoles as imidazoline I<sub>2</sub> receptor ligands for Alzheimer's disease.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 1 | 9.92 | 9.92 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4861277 | — | — | 1 | 9.92 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4861277 | — | Ki | = | 0.1202 | nM | 9.92 |