Assay Detail
Binding
CHEMBL4828242
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Binding affinity to BRD9 (unknown origin) by BROMOscan method
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
New Design Rules for Developing Potent Cell-Active Inhibitors of the Nucleosome Remodeling Factor (NURF) via BPTF Bromodomain Inhibition.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Kd | 3 | 8.53 | 9.62 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4861491 | — | — | 1 | 9.62 |
| CHEMBL4872300 | — | — | 1 | 9.33 |
| CHEMBL4848701 | — | — | 1 | 6.64 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4861491 | — | Kd | = | 0.24 | nM | 9.62 |
| CHEMBL4872300 | — | Kd | = | 0.47 | nM | 9.33 |
| CHEMBL4848701 | — | Kd | = | 230.0 | nM | 6.64 |