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Assay Detail

CHEMBL4828891

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antileishmanial activity against Leishmania amazonensis (MHOM/BR/73/M2269) promastigotes assessed as inhibition of parasite growth measured after 24 hrs by MTT assay
4
Total Activities
4
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Leishmania amazonensis
Confidence 1 — Organism
Curated By Autocuration

Target

Leishmania amazonensis (CHEMBL612877)
Type ORGANISM
Organism Leishmania amazonensis

Publication

Mechanistic Insights into the Leishmanicidal and Bactericidal Activities of Batroxicidin, a Cathelicidin-Related Peptide from a South American Viper (<i>Bothrops atrox</i>).
Dematei A, Nunes JB, Moreira DC, Jesus JA, Laurenti MD, Mengarda ACA, Vieira MS, do Amaral CP, Domingues MM, de Moraes J, Passero LFD, Brand G, Bessa LJ, Wimmer R, Kuckelhaus SAS, Tomás AM, Santos NC, Plácido A, Eaton P, Leite JRSA.
J Nat Prod (2021) 84 : 1787 -1798
PubMed 34077221 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 4 5.79 7.62

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL267345 AMPHOTERICIN B 4.0 1 7.62
CHEMBL4861276 1 5.31
CHEMBL4864681 1 5.17
CHEMBL4846717 1 5.05

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL267345 AMPHOTERICIN B EC50 = 24.0 nM 7.62
CHEMBL4861276 EC50 = 4900.0 nM 5.31
CHEMBL4864681 EC50 = 6740.0 nM 5.17
CHEMBL4846717 EC50 = 8860.0 nM 5.05