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Assay Detail

CHEMBL4832359

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Binding
Inhibition of KDM4D (unknown origin)
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Lysine-specific demethylase 4D (CHEMBL6138)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Discovery of a potent and selective inhibitor of histone lysine demethylase KDM4D.
Fang Z, Liu Y, Zhang R, Chen Q, Wang T, Yang W, Fan Y, Yu C, Xiang R, Yang S.
Eur J Med Chem (2021) 223 : 113662 -113662
PubMed 34237635 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 6.54 6.54

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL1982368 1 6.54

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL1982368 IC50 = 290.0 nM 6.54