Assay Detail
Functional
CHEMBL4833084
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Suppression of IL-17A production in human Th17 cells incubated for 4 days by IL-17 HTRF assay
48
Total Activities
48
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | Th17 |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
AZD0284, a Potent, Selective, and Orally Bioavailable Inverse Agonist of Retinoic Acid Receptor-Related Orphan Receptor C2.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 48 | 7.38 | 8.22 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4852138 | — | — | 1 | 8.22 |
| CHEMBL4859385 | — | — | 1 | 8.15 |
| CHEMBL4877500 | — | — | 1 | 8.15 |
| CHEMBL4864990 | — | — | 1 | 8.15 |
| CHEMBL4865776 | — | — | 1 | 8.00 |
| CHEMBL4864604 | — | — | 1 | 7.96 |
| CHEMBL4868864 | — | — | 1 | 7.96 |
| CHEMBL4866908 | — | — | 1 | 7.96 |
| CHEMBL4853971 | — | — | 1 | 7.92 |
| CHEMBL4875842 | — | — | 1 | 7.85 |
| CHEMBL4864731 | — | — | 1 | 7.82 |
| CHEMBL4850055 | — | — | 1 | 7.77 |
| CHEMBL4847308 | — | — | 1 | 7.70 |
| CHEMBL4849302 | — | — | 1 | 7.70 |
| CHEMBL4855387 | — | — | 1 | 7.66 |
| CHEMBL4848388 | — | — | 1 | 7.64 |
| CHEMBL4865352 | — | — | 1 | 7.58 |
| CHEMBL4866227 | — | — | 1 | 7.55 |
| CHEMBL4857284 | — | — | 1 | 7.54 |
| CHEMBL4562895 | — | — | 1 | 7.52 |
| CHEMBL4463668 | — | — | 1 | 7.52 |
| CHEMBL4846059 | — | — | 1 | 7.51 |
| CHEMBL4865573 | — | — | 1 | 7.51 |
| CHEMBL4856430 | — | — | 1 | 7.48 |
| CHEMBL4870856 | — | — | 1 | 7.41 |
| CHEMBL4862137 | — | — | 1 | 7.33 |
| CHEMBL4876902 | — | — | 1 | 7.27 |
| CHEMBL4868619 | — | — | 1 | 7.24 |
| CHEMBL4857395 | — | — | 1 | 7.24 |
| CHEMBL4875667 | — | — | 1 | 7.22 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4852138 | — | IC50 | = | 6.0 | nM | 8.22 |
| CHEMBL4859385 | — | IC50 | = | 7.0 | nM | 8.15 |
| CHEMBL4864990 | — | IC50 | = | 7.0 | nM | 8.15 |
| CHEMBL4877500 | — | IC50 | = | 7.0 | nM | 8.15 |
| CHEMBL4865776 | — | IC50 | = | 10.0 | nM | 8.00 |
| CHEMBL4864604 | — | IC50 | = | 11.0 | nM | 7.96 |
| CHEMBL4868864 | — | IC50 | = | 11.0 | nM | 7.96 |
| CHEMBL4866908 | — | IC50 | = | 11.0 | nM | 7.96 |
| CHEMBL4853971 | — | IC50 | = | 12.0 | nM | 7.92 |
| CHEMBL4875842 | — | IC50 | = | 14.0 | nM | 7.85 |
| CHEMBL4864731 | — | IC50 | = | 15.0 | nM | 7.82 |
| CHEMBL4850055 | — | IC50 | = | 17.0 | nM | 7.77 |
| CHEMBL4847308 | — | IC50 | = | 20.0 | nM | 7.70 |
| CHEMBL4849302 | — | IC50 | = | 20.0 | nM | 7.70 |
| CHEMBL4855387 | — | IC50 | = | 22.0 | nM | 7.66 |
| CHEMBL4848388 | — | IC50 | = | 23.0 | nM | 7.64 |
| CHEMBL4865352 | — | IC50 | = | 26.0 | nM | 7.58 |
| CHEMBL4866227 | — | IC50 | = | 28.0 | nM | 7.55 |
| CHEMBL4857284 | — | IC50 | = | 29.0 | nM | 7.54 |
| CHEMBL4562895 | — | IC50 | = | 30.0 | nM | 7.52 |
| CHEMBL4463668 | — | IC50 | = | 30.0 | nM | 7.52 |
| CHEMBL4846059 | — | IC50 | = | 31.0 | nM | 7.51 |
| CHEMBL4865573 | — | IC50 | = | 31.0 | nM | 7.51 |
| CHEMBL4856430 | — | IC50 | = | 33.0 | nM | 7.48 |
| CHEMBL4870856 | — | IC50 | = | 39.0 | nM | 7.41 |
| CHEMBL4862137 | — | IC50 | = | 47.0 | nM | 7.33 |
| CHEMBL4876902 | — | IC50 | = | 54.0 | nM | 7.27 |
| CHEMBL4868619 | — | IC50 | = | 57.0 | nM | 7.24 |
| CHEMBL4857395 | — | IC50 | = | 58.0 | nM | 7.24 |
| CHEMBL4875667 | — | IC50 | = | 60.0 | nM | 7.22 |
| CHEMBL4847134 | — | IC50 | = | 63.0 | nM | 7.20 |
| CHEMBL4870339 | — | IC50 | = | 72.0 | nM | 7.14 |
| CHEMBL4850359 | — | IC50 | = | 77.0 | nM | 7.11 |
| CHEMBL4870686 | — | IC50 | = | 86.0 | nM | 7.07 |
| CHEMBL4868403 | — | IC50 | = | 91.0 | nM | 7.04 |
| CHEMBL4853746 | — | IC50 | = | 102.0 | nM | 6.99 |
| CHEMBL4856963 | — | IC50 | = | 102.0 | nM | 6.99 |
| CHEMBL4854122 | — | IC50 | = | 115.0 | nM | 6.94 |
| CHEMBL4872141 | — | IC50 | = | 120.0 | nM | 6.92 |
| CHEMBL4847761 | — | IC50 | = | 127.0 | nM | 6.90 |
| CHEMBL4878173 | — | IC50 | = | 158.0 | nM | 6.80 |
| CHEMBL4845714 | — | IC50 | = | 224.0 | nM | 6.65 |
| CHEMBL4855766 | — | IC50 | = | 248.0 | nM | 6.61 |
| CHEMBL4868767 | — | IC50 | = | 286.0 | nM | 6.54 |
| CHEMBL4869175 | — | IC50 | = | 287.0 | nM | 6.54 |
| CHEMBL4852181 | — | IC50 | = | 360.0 | nM | 6.44 |
| CHEMBL4875795 | — | IC50 | = | 423.0 | nM | 6.37 |
| CHEMBL4856950 | — | IC50 | > | 3330.0 | nM | - |