Assay Detail
Binding
CHEMBL4834053
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Binding affinity to human serum albumin by fluorescence polarization assay
22
Total Activities
22
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Identification and Validation of New Interleukin-2 Ligands Using DNA-Encoded Libraries.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Kd | 22 | 6.26 | 7.70 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4874500 | — | — | 1 | 7.70 |
| CHEMBL4875916 | — | — | 1 | 7.52 |
| CHEMBL4852232 | — | — | 1 | 7.16 |
| CHEMBL4845813 | — | — | 1 | 6.77 |
| CHEMBL4870031 | — | — | 1 | 6.68 |
| CHEMBL4866037 | — | — | 1 | 6.66 |
| CHEMBL4866759 | — | — | 1 | 6.57 |
| CHEMBL4877313 | — | — | 1 | 6.54 |
| CHEMBL4856339 | — | — | 1 | 6.51 |
| CHEMBL4869829 | — | — | 1 | 6.41 |
| CHEMBL4879282 | — | — | 1 | 6.37 |
| CHEMBL4873867 | — | — | 1 | 6.24 |
| CHEMBL4855828 | — | — | 1 | 6.11 |
| CHEMBL4870525 | — | — | 1 | 6.09 |
| CHEMBL4863588 | — | — | 1 | 6.00 |
| CHEMBL4876740 | — | — | 1 | 5.82 |
| CHEMBL4872601 | — | — | 1 | 5.77 |
| CHEMBL4851618 | — | — | 1 | 5.70 |
| CHEMBL4861027 | — | — | 1 | 5.48 |
| CHEMBL4867370 | — | — | 1 | 5.40 |
| CHEMBL4871406 | — | — | 1 | 5.14 |
| CHEMBL4846246 | — | — | 1 | 5.02 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4874500 | — | Kd | = | 20.0 | nM | 7.70 |
| CHEMBL4875916 | — | Kd | = | 30.0 | nM | 7.52 |
| CHEMBL4852232 | — | Kd | = | 70.0 | nM | 7.16 |
| CHEMBL4845813 | — | Kd | = | 170.0 | nM | 6.77 |
| CHEMBL4870031 | — | Kd | = | 210.0 | nM | 6.68 |
| CHEMBL4866037 | — | Kd | = | 220.0 | nM | 6.66 |
| CHEMBL4866759 | — | Kd | = | 270.0 | nM | 6.57 |
| CHEMBL4877313 | — | Kd | = | 290.0 | nM | 6.54 |
| CHEMBL4856339 | — | Kd | = | 310.0 | nM | 6.51 |
| CHEMBL4869829 | — | Kd | = | 390.0 | nM | 6.41 |
| CHEMBL4879282 | — | Kd | = | 430.0 | nM | 6.37 |
| CHEMBL4873867 | — | Kd | = | 580.0 | nM | 6.24 |
| CHEMBL4855828 | — | Kd | = | 780.0 | nM | 6.11 |
| CHEMBL4870525 | — | Kd | = | 820.0 | nM | 6.09 |
| CHEMBL4863588 | — | Kd | = | 1000.0 | nM | 6.00 |
| CHEMBL4876740 | — | Kd | = | 1500.0 | nM | 5.82 |
| CHEMBL4872601 | — | Kd | = | 1700.0 | nM | 5.77 |
| CHEMBL4851618 | — | Kd | = | 2000.0 | nM | 5.70 |
| CHEMBL4861027 | — | Kd | = | 3300.0 | nM | 5.48 |
| CHEMBL4867370 | — | Kd | = | 4000.0 | nM | 5.40 |
| CHEMBL4871406 | — | Kd | = | 7200.0 | nM | 5.14 |
| CHEMBL4846246 | — | Kd | = | 9600.0 | nM | 5.02 |