Assay Detail
Binding
CHEMBL4839004
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Displacement of [3H]-PSB15900 from human platelet membrane Gq incubated for 90 mins by scintillation counter method
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Cell Type | Platelet |
| Subcellular | Membrane |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Feature-Based Molecular Networking for the Targeted Identification of G<sub>q</sub>-Inhibiting FR900359 Derivatives.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 2 | 8.08 | 8.66 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4171381 | — | — | 1 | 8.66 |
| CHEMBL4873047 | — | — | 1 | 7.50 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4171381 | — | Ki | = | 2.188 | nM | 8.66 |
| CHEMBL4873047 | — | Ki | = | 31.62 | nM | 7.50 |