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Assay Detail

CHEMBL4840219

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antimalarial activity against asexual late stage (IV-V) Plasmodium falciparum 3D7 gametocytes expressing CBG99 luciferase infected in human red blood cells assessed as reduction in gametocyte viability measured after 72 hrs by luminescence based assay
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Plasmodium falciparum
Confidence 1 — Organism
Curated By Autocuration

Target

Plasmodium falciparum (CHEMBL364)
Type ORGANISM
Organism Plasmodium falciparum

Publication

Development of Potent 3-Br-isoxazoline-Based Antimalarial and Antileishmanial Compounds.
Galbiati A, Zana A, Coser C, Tamborini L, Basilico N, Parapini S, Taramelli D, Conti P.
ACS Med Chem Lett (2021) 12 : 1726 -1732
PubMed 34795860 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 4.98 4.98

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL4854616 1 4.98

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL4854616 IC50 = 10400.0 nM 4.98