Assay Detail
Binding
CHEMBL4840832
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Displacement of [3H]CP55940 from human CB1 receptor transfected in CHO cells measured for 1.5 hrs by liquid scintillation counting analysis
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Cell Type | CHO |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Δ<sup>9</sup>-<i>cis</i>-Tetrahydrocannabinol: Natural Occurrence, Chirality, and Pharmacology.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 3 | 6.61 | 7.66 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL465 | DRONABINOL | 4.0 | 1 | 7.66 |
| CHEMBL4845760 | — | — | 1 | 6.64 |
| CHEMBL4862731 | — | — | 1 | 5.54 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL465 | DRONABINOL | Ki | = | 22.0 | nM | 7.66 |
| CHEMBL4845760 | — | Ki | = | 228.0 | nM | 6.64 |
| CHEMBL4862731 | — | Ki | = | 2900.0 | nM | 5.54 |