Assay Detail
Binding
CHEMBL4843290
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Inhibition of human ERG expressed in CHO by QPatch assay
11
Total Activities
11
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Cell Type | CHO |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Voltage-gated inwardly rectifying potassium channel KCNH2 (CHEMBL240) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
Discovery of IACS-9779 and IACS-70465 as Potent Inhibitors Targeting Indoleamine 2,3-Dioxygenase 1 (IDO1) Apoenzyme.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 11 | 5.26 | 6.13 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4846783 | — | — | 1 | 6.13 |
| CHEMBL4853672 | — | — | 1 | 5.85 |
| CHEMBL4870418 | — | — | 1 | 5.68 |
| CHEMBL4848514 | — | — | 1 | 5.25 |
| CHEMBL4859064 | — | — | 1 | 5.00 |
| CHEMBL4861332 | — | — | 1 | 4.96 |
| CHEMBL4845961 | — | — | 1 | 4.92 |
| CHEMBL4871068 | — | — | 1 | 4.85 |
| CHEMBL4864639 | — | — | 1 | 4.68 |
| CHEMBL4863359 | — | — | 1 | - |
| CHEMBL4849414 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4846783 | — | IC50 | = | 740.0 | nM | 6.13 |
| CHEMBL4853672 | — | IC50 | = | 1400.0 | nM | 5.85 |
| CHEMBL4870418 | — | IC50 | = | 2100.0 | nM | 5.68 |
| CHEMBL4848514 | — | IC50 | = | 5600.0 | nM | 5.25 |
| CHEMBL4859064 | — | IC50 | = | 9900.0 | nM | 5.00 |
| CHEMBL4861332 | — | IC50 | = | 11000.0 | nM | 4.96 |
| CHEMBL4845961 | — | IC50 | = | 12000.0 | nM | 4.92 |
| CHEMBL4871068 | — | IC50 | = | 14000.0 | nM | 4.85 |
| CHEMBL4864639 | — | IC50 | = | 21000.0 | nM | 4.68 |
| CHEMBL4863359 | — | IC50 | > | 30000.0 | nM | - |
| CHEMBL4849414 | — | IC50 | > | 30000.0 | nM | - |