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Assay Detail

CHEMBL4844512

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of electric eel AChE using acetylthiocholine iodide as substrate incubated for 5 mins followed by substrate addition and measured after 5 mins by spectrophotometric based Ellman's method
21
Total Activities
21
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Electrophorus electricus
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Acetylcholinesterase (CHEMBL4078)
Type SINGLE PROTEIN
Organism Electrophorus electricus

Publication

Discovery of 1-(phenylsulfonyl)-1H-indole-based multifunctional ligands targeting cholinesterases and 5-HT<sub>6</sub> receptor with anti-aggregation properties against amyloid-beta and tau.
Wichur T, Pasieka A, Godyń J, Panek D, Góral I, Latacz G, Honkisz-Orzechowska E, Bucki A, Siwek A, Głuch-Lutwin M, Knez D, Brazzolotto X, Gobec S, Kołaczkowski M, Sabate R, Malawska B, Więckowska A.
Eur J Med Chem (2021) 225 : 113783 -113783
PubMed 34461507 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 21 6.85 8.07

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL4850546 1 8.07
CHEMBL502 DONEPEZIL 4.0 1 7.96
CHEMBL4850051 1 7.68
CHEMBL95 TACRINE 4.0 1 7.64
CHEMBL4874513 1 7.24
CHEMBL4877482 1 7.14
CHEMBL4848231 1 6.52
CHEMBL4878361 1 5.54
CHEMBL4878383 1 5.37
CHEMBL4847532 1 5.32
CHEMBL4866788 1 -
CHEMBL4850488 1 -
CHEMBL4845823 1 -
CHEMBL4854972 1 -
CHEMBL4864206 1 -
CHEMBL4868597 1 -
CHEMBL4851595 1 -
CHEMBL4852099 1 -
CHEMBL4847373 1 -
CHEMBL4863218 1 -
CHEMBL4871964 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL4850546 IC50 = 8.42 nM 8.07
CHEMBL502 DONEPEZIL IC50 = 11.0 nM 7.96
CHEMBL4850051 IC50 = 20.9 nM 7.68
CHEMBL95 TACRINE IC50 = 23.0 nM 7.64
CHEMBL4874513 IC50 = 57.54 nM 7.24
CHEMBL4877482 IC50 = 72.48 nM 7.14
CHEMBL4848231 IC50 = 303.1 nM 6.52
CHEMBL4878361 IC50 = 2869.0 nM 5.54
CHEMBL4878383 IC50 = 4236.0 nM 5.37
CHEMBL4847532 IC50 = 4841.0 nM 5.32
CHEMBL4866788 IC50 - -
CHEMBL4850488 IC50 - -
CHEMBL4845823 IC50 - -
CHEMBL4854972 IC50 - -
CHEMBL4864206 IC50 = 4467000.0 nM -
CHEMBL4868597 IC50 - -
CHEMBL4851595 IC50 - -
CHEMBL4852099 IC50 = 6214000.0 nM -
CHEMBL4847373 IC50 - -
CHEMBL4863218 IC50 - -
CHEMBL4871964 IC50 - -