Assay Detail
Binding
CHEMBL4880317
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Radioligand assay (DRD4.4)
1
Total Activities
1
Compounds Tested
1
Activity Types
2
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Data for DCP probe ABT-724
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 1 | 7.20 | 7.20 |
Assay Parameters
| Parameter | Type | Value | Units | Text |
|---|---|---|---|---|
| Assay publication | Assay publication | - | — | PMID: 15087502 |
| Target protein type | Target protein type | - | — | Membrane preparations expressing the human D4 variants |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL440687 | ABT-724 | — | 1 | 7.20 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL440687 | ABT-724 | Ki | = | 63.6 | nM | 7.20 |