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Assay Detail

CHEMBL4880938

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Binding
Cellular luciferase reporter assay using the SN12C-MEF2-luc cell line and ONE-Glo
2
Total Activities
2
Compounds Tested
1
Activity Types
1
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Cell Type SN12C
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Mitogen-activated protein kinase 7 (CHEMBL5332)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Data for DCP probe BAY-885
SGC Frankfurt
(2021)
· DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 2 5.95 6.94

Assay Parameters

Parameter Type Value Units Text
Assay publication Assay publication - PMID: 30563338

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL4445670 BAY-885 1 6.94
CHEMBL4455582 BAY-693 1 4.96

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL4445670 BAY-885 IC50 = 115.0 nM 6.94
CHEMBL4455582 BAY-693 IC50 = 11000.0 nM 4.96