Assay Detail
Binding
CHEMBL4882233
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Ca flux
2
Total Activities
2
Compounds Tested
1
Activity Types
1
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Data for DCP probe BI 639667
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 7.62 | 7.62 |
Assay Parameters
| Parameter | Type | Value | Units | Text |
|---|---|---|---|---|
| Additional information | Additional information | - | — | CCR1 molecular potency |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4456123 | BI 639667 | 1.0 | 1 | 7.62 |
| CHEMBL4539555 | BI 9307 | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4456123 | BI 639667 | IC50 | = | 24.0 | nM | 7.62 |
| CHEMBL4539555 | BI 9307 | IC50 | > | 3000.0 | nM | - |