Assay Detail

CHEMBL4883191

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional

CHO-based cAMP assay (mouse)

ChEMBL ↗

Free Research Context This assay will appear in recent viewed items on this browser. Open the demo workspace to preview project-only review queues.

Research home Demo workspace

Target

G-protein coupled receptor 52 (CHEMBL4105791) ↗

Open DB target context

Use one target anchor to keep assay intent, target linkage, and tested compound review aligned.

Loading context

G-protein coupled receptor 52 (CHEMBL4105791) is the working anchor for this assay review. Loading the live Open DB target snapshot…

Primary target G-protein coupled receptor 52

CHEMBL4105791

Anchored from Assay target.

Protein identity G-protein coupled receptor 52

Disease frame Disease evidence pending

Open the live target snapshot or evidence card before reviewing assay metadata so target fit and disease framing stay reusable.

Review focus Open DB context pending

Open the live target snapshot before relying on this target frame across surface handoff.

Open target snapshot Open evidence card Search with this context

Total Activities

Compounds Tested

Activity Types

Assay Parameters

Assay Information

Assay Type	Functional
Organism	Mus musculus
Confidence	9 — Direct single protein target
Curated By	Autocuration

Target

G-protein coupled receptor 52 (CHEMBL4105791) ↗

Type	SINGLE PROTEIN
Organism	Mus musculus

Publication

Data for DCP probe TP-024

SGC Frankfurt
(2021)
· DOI

Activity Statistics

Type	Count	Avg pChEMBL	Best pChEMBL
EC50	1	6.85	6.85

Assay Parameters

Parameter	Type	Value	Units	Text
Target protein type	Target protein type	-	—	GPR52 expressed CHO cell line

Compounds Tested

Compound	Name	Phase	Activities	Best pChEMBL
CHEMBL4082756	TP-024	—	1	6.85

Activity Data

Compound	Name	Type	Rel.	Value	Units	pChEMBL
CHEMBL4082756	TP-024	EC50	=	141.0	nM	6.85