Assay Detail
Binding
CHEMBL4883205
Review assay metadata, readout intent, target linkage, and publication context from the same page.
NanoBRET (SGC Frankfurt) (DYRK1A)
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Dual specificity tyrosine-phosphorylation-regulated kinase 1A (CHEMBL2292) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
Data for DCP probe T3-CLK
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 7.50 | 7.50 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4531334 | T3-CLK | — | 1 | 7.50 |
| CHEMBL4576555 | T3-CLK-N | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4531334 | T3-CLK | IC50 | = | 32.0 | nM | 7.50 |
| CHEMBL4576555 | T3-CLK-N | IC50 | > | 10000.0 | nM | - |