Assay Detail

CHEMBL4883299

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Binding

BRET-Gi dissociation assay

ChEMBL ↗

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Target

D(4) dopamine receptor (CHEMBL219) ↗

Open DB target context

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D(4) dopamine receptor (CHEMBL219) is the working anchor for this assay review. Loading the live Open DB target snapshot…

Primary target D(4) dopamine receptor

CHEMBL219

Anchored from Assay target.

Protein identity D(4) dopamine receptor

Disease frame Disease evidence pending

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Review focus Open DB context pending

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Total Activities

Compounds Tested

Activity Types

Assay Parameters

Assay Information

Assay Type	Binding
Organism	Homo sapiens
Confidence	9 — Direct single protein target
Curated By	Autocuration

Target

D(4) dopamine receptor (CHEMBL219) ↗

Type	SINGLE PROTEIN
Organism	Homo sapiens

Publication

Data for DCP probe UCSF924

SGC Frankfurt
(2021)
· DOI

Activity Statistics

Type	Count	Avg pChEMBL	Best pChEMBL
EC50	1	9.70	9.70

Assay Parameters

Parameter	Type	Value	Units	Text
Assay publication	Assay publication	-	—	PMID: 29051383

Compounds Tested

Compound	Name	Phase	Activities	Best pChEMBL
CHEMBL3480577	UCSF924	—	1	9.70

Activity Data

Compound	Name	Type	Rel.	Value	Units	pChEMBL
CHEMBL3480577	UCSF924	EC50	=	0.2	nM	9.70