Skip to main content
Free research Free research Free assay review with research home and workspace preview
Quick search ChEMBL 36
Assay Detail

CHEMBL4885811

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
BRD3 BD2 Bromoscan (DiscoverX)
1
Total Activities
1
Compounds Tested
1
Activity Types
2
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Bromodomain-containing protein 3 (CHEMBL1795186)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Data for DCP probe GSK620
SGC Frankfurt
(2021)
· DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Kd 1 7.90 7.90

Assay Parameters

Parameter Type Value Units Text
Assay publication Assay publication - PMID: 32702236
Target protein length Target protein length - BD2

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL4635134 GSK620 1 7.90

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL4635134 GSK620 Kd = 12.59 nM 7.90