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Assay Detail

CHEMBL4886126

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Fluorescence Cross Correlation Spectroscopy (FCCS) mouse
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Mus musculus
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Monocarboxylate transporter 4 (CHEMBL4802065)
Type SINGLE PROTEIN
Organism Mus musculus

Publication

Data for DCP probe MSC-4381
SGC Frankfurt
(2021)
· DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 1 6.60 6.60

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL4802043 MSC-4381 1 6.60

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL4802043 MSC-4381 Ki = 252.0 nM 6.60