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Assay Detail

CHEMBL4886403

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
hPDE4D3 PDE scan
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

3',5'-cyclic-AMP phosphodiesterase 4D (CHEMBL288)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Data for DCP probe JNJ-42396302
SGC Frankfurt
(2021)
· DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 1 4.82 4.82

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL2180408 JNJ-42396302 1.0 1 4.82

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL2180408 JNJ-42396302 Ki = 15000.0 nM 4.82