Assay Detail
Binding
CHEMBL4888385
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PPARgamma In-house nuclear receptor screen
2
Total Activities
1
Compounds Tested
2
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Peroxisome proliferator-activated receptor gamma (CHEMBL235) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
Data for DCP probe JNJ-54119936
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Inhibition | 1 | - | - |
| IC50 | 1 | 5.27 | 5.27 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4802042 | JNJ-54119936 | — | 2 | 5.27 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4802042 | JNJ-54119936 | IC50 | = | 5400.0 | nM | 5.27 |
| CHEMBL4802042 | JNJ-54119936 | Inhibition | = | 28.2 | % | - |