Assay Detail
Binding
CHEMBL5029280
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of mammalian Alpha-glucosidase (unknown origin) using PNPG as substrate pretreated for 20 mins followed by substrate addition measured after 26 mins
4
Total Activities
2
Compounds Tested
2
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Positional Isomeric Effects on the Optical Properties, Multivalent Glycosidase Inhibition Effect, and Hypoglycemic Effect of Perylene Bisimide-deoxynojirimycin Conjugates.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Inhibition | 2 | - | - |
| IC50 | 2 | 4.89 | 4.93 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5078012 | — | — | 2 | 4.93 |
| CHEMBL5090920 | — | — | 2 | 4.84 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5078012 | — | IC50 | = | 11610.0 | nM | 4.93 |
| CHEMBL5090920 | — | IC50 | = | 14420.0 | nM | 4.84 |
| CHEMBL5078012 | — | Inhibition | - | % | - | |
| CHEMBL5090920 | — | Inhibition | - | % | - |